BDBM25150 (2E)-N-hydroxy-3-[3-(phenylsulfamoyl)phenyl]prop-2-enamide::Belinosta::Belinostat::PXD-101::PXD101
SMILES ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)Nc1ccccc1
InChI Key InChIKey=NCNRHFGMJRPRSK-MDZDMXLPSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 25150
Affinity DataKi: 51nMAssay Description:Competitive inhibition of HDAC7 using KI-104 as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibition of human HDAC7More data for this Ligand-Target Pair
Affinity DataIC50: 598nMAssay Description:Antagonistic affinity measured as pA2 value on 5-hydroxytryptamine 2B receptor of the rat stomach fundusMore data for this Ligand-Target Pair
Affinity DataEC50: 67nMAssay Description:Inhibition of recombinant human HDAC7 expressed in baculovirus expression system using KI-104 as substrate incubated for 3 hrs by by fluorescence-bas...More data for this Ligand-Target Pair